Turinabol

Posted by: @thecaptn

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Is 50mg a worthwhile dose? Reason being I can get 50mg caps.

If your getting authentic t-bol 50mg a day is plenty as a starting point....imho.

Studies show that 10mg a day will compete for shbg allowing for more free test in your bloodstream.

Most bros I have spoken with about t-bol agree that 50mg a day should be plenty for mid-level experienced Bros for putting on some lean mass.

For beginners I would recommend 30-40 mgs a day to see how you react. If you have 50mg caps and have not used t-bol before or in any case for that matter you want to drink plenty of water, use taurine, and potassium to prevent locking up your muscles. You should be at least drinking plenty of water while using ANY orals anyways.

I openly admit I do not know at what dose we would encounter the point of diminishing returns?

Anyone?

Disposition and excretion of the anabolic steroid Oral-Turinabol (1;4-chloro-17 alpha-methyl-androsta-1,4-diene-17 beta-hydroxy-3-one) were investigated in male volunteers. Following single p.o. and i.v. administration of the tritium-labelled compound the plasma concentration courses of total radioactivity (1 and 1-metabolites) and of the unchanged parent drug as well as the urinary excretion were estimated. From these data model independent pharmacokinetic parameters based on statistical moments were calculated. 1 is almost completely absorbed after p.o. administration of 10 mg per volunteer. Peak concentrations of total radioactivity and of 1 in plasma were reached about 3 h p.a. Irregularities observed in the plasma level profile following both p.o. and i.v. administration of 1 are due to a marked enterohepatic circulation. Orally given 1 is subject to a first-pass effect, resulting in a diminished systematic availability. The AUC-ratio of the unchanged drug and the total radioactivity of 1 : 13 shows the predominance of metabolites in plasma. After i.v. administration the disposition of unchanged 1 was found biphasically with a terminal half-life of 16 h. 1 and its metabolites are preferentially excreted via the kidneys. The urinary total radioactivity represented about 60% of the dose following both administrations.

Due to its affinity to SHBG 1 is able to compete for the protein binding of testosterone, resulting in an increased plasma level of non protein-bound testosterone.

LM1

good post 👍

Posted by: @liquidmuscle1

↑

If your getting authentic t-bol 50mg a day is plenty as a starting point....imho.

Studies show that 10mg a day will compete for shbg allowing for more free test in your bloodstream.

Most bros I have spoken with about t-bol agree that 50mg a day should be plenty for mid-level experienced Bros for putting on some lean mass.

For beginners I would recommend 30-40 mgs a day to see how you react. If you have 50mg caps and have not used t-bol before or in any case for that matter you want to drink plenty of water, use taurine, and potassium to prevent locking up your muscles. You should be at least drinking plenty of water while using ANY orals anyways.

I openly admit I do not know at what dose we would encounter the point of diminishing returns?

Anyone?

Disposition and excretion of the anabolic steroid Oral-Turinabol (1;4-chloro-17 alpha-methyl-androsta-1,4-diene-17 beta-hydroxy-3-one) were investigated in male volunteers. Following single p.o. and i.v. administration of the tritium-labelled compound the plasma concentration courses of total radioactivity (1 and 1-metabolites) and of the unchanged parent drug as well as the urinary excretion were estimated. From these data model independent pharmacokinetic parameters based on statistical moments were calculated. 1 is almost completely absorbed after p.o. administration of 10 mg per volunteer. Peak concentrations of total radioactivity and of 1 in plasma were reached about 3 h p.a. Irregularities observed in the plasma level profile following both p.o. and i.v. administration of 1 are due to a marked enterohepatic circulation. Orally given 1 is subject to a first-pass effect, resulting in a diminished systematic availability. The AUC-ratio of the unchanged drug and the total radioactivity of 1 : 13 shows the predominance of metabolites in plasma. After i.v. administration the disposition of unchanged 1 was found biphasically with a terminal half-life of 16 h. 1 and its metabolites are preferentially excreted via the kidneys. The urinary total radioactivity represented about 60% of the dose following both administrations.

Due to its affinity to SHBG 1 is able to compete for the protein binding of testosterone, resulting in an increased plasma level of non protein-bound testosterone.

LM1